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Umbralisib hydrochloride
😃Good
Catalog No. T17066Cas No. 1532533-78-0
Alias TGR-1202 hydrochloride, RP5264 hydrochloride
Umbralisib hydrochloride is a novel PI3Kδ inhibitor (IC50 and EC50 of 22.2 nM and 24.3 nM, respectively). Umbralisib hydrochloride is also active against CK1ε (EC50: 6.0 μM).
Umbralisib hydrochloride
😃Good
Catalog No. T17066Alias TGR-1202 hydrochloride, RP5264 hydrochlorideCas No. 1532533-78-0
Umbralisib hydrochloride is a novel PI3Kδ inhibitor (IC50 and EC50 of 22.2 nM and 24.3 nM, respectively). Umbralisib hydrochloride is also active against CK1ε (EC50: 6.0 μM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $53 | 5 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Umbralisib hydrochloride is a novel PI3Kδ inhibitor (IC50 and EC50 of 22.2 nM and 24.3 nM, respectively). Umbralisib hydrochloride is also active against CK1ε (EC50: 6.0 μM). |
| Targets&IC50 | PI3Kδ:22.2 nM |
| Alias | TGR-1202 hydrochloride, RP5264 hydrochloride |
| Molecular Weight | 608.01 |
| Formula | C31H25ClF3N5O3 |
| Cas No. | 1532533-78-0 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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